R03AC03 - Terbutaline |
Not porphyrinogenic |
NP |
Rationale
Probably non-CYP metabolism. One reference: authorised. Significant clinical experience of non-porphyrinogenicity.
Chemical description
Adrenergic used in asthma administered in inhalation aerosol (5mg x 4) in asthma. Metabolised by sulfatation and excreted in urine in conjugated form. No clinical data pointing to CYP-interaction.
Personal communication
Andersson C, patient reports: tolerated (n=11).
Used in porphyria ward (Sweden).
IPNet drug reports
Uneventful use reported in 20 patients with acute porphyria.
Similar drugs
References
| # | Citation details | PubMed ID |
|---|---|---|
| Porphyria Drug Lists | ||
| 1. | French List
Centre Français des Porphyries
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Tradenames